MLN-4760 is a novel, potent and selective human angiotensin-converting (ACE2) inhibitor with IC50 of 0.44 nM and with excellent selectivity (>5000-fold) versus related enzymes including human testicular ACE (IC50, >100 μM) and bovine carboxypeptidase A (CPDA; IC50, 27 μM). In huMNCs, MLN-4760-B detected 63% ACE2 with 28-fold selectivity over ACE.
纯度:≥98%
CAS:305335-31-3