Peripheral HH1R antagonist
CAS：79794-75-5
分子式：C22H23ClN2O2
分子量：382.88
纯度：98%
存储：Store at -20°C

Background:

Loratadine(SCH-29851) is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.IC50 value: 32 uMTarget: H1-receptorLoratadine is a non-sedative antihistamine that inhibits histamine-induced activities of IL-6 and IL-8 secretion in endothelial cells.

参考文献:
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