α1adrenoceptor-MO-1是一种S型对映体,对alpha1adrenergicreceptor具有亲和性,可以抗α-肾上腺素能,同时能够止痛;比R型对映体的活性高。
CAS:161905-64-2
分子式:C20H24ClN5O
分子量:385.89
纯度:98%
存储:Store at -20°C
Background:
α1 adrenoceptor-MO-1, an S enantiomer, has affinity at alpha 1 adrenergic receptor, shows alphalytic activity, and possesses analgesic action; more active than R enantiomer.
α1 adrenoceptor-MO-1 (the S enantiomer) and R enantiomer are more active than the corresponding racemates, but α1 adrenoceptor-MO-1 is more active than R enantiomer[1].
[1]. Pharmacologically active enantiomers. WO 1995001354 A1