Levetimide 是一种有效的立体选择性 [3H](+)pentazocine 结合抑制剂，Ki 为 2.2 nM。
CAS：21888-99-3
分子式：C23H26N2O2
分子量：362.46
纯度：98%
存储：Store at -20°C

Background:

Levetimide is a potent and stereoselective inhibitor of [3H](+)pentazocine binding, with a Ki of 2.2 nM[1].

Levetimide potently inhibits [3H]DTG binding although without stereoselectivity (Ki value of 103 nM) [1].

[1]. DeHaven-Hudkins DL, et al. Binding of dexetimide and levetimide to [3H](+)pentazocine- and [3H]1,3-di(2-tolyl)guanidine-defined sigma recognition sites. Life Sci. 1991;49(18):PL135-9.