CGRPantagonist1是高效的CGRP受体拮抗剂,Ki和IC50值分别为35和57nM。
货号:ajcx12494
CAS:1123757-49-2
分子式:C29H26N4O4
分子量:494.54
溶解度:Soluble in DMSO
纯度:98%
存储:Store at -20°C
库存:
现货Background:
CGRP antagonist 1 is a highly potent CGRP receptor antagonist with a Ki and IC50 of 35 and 57 nM, respectively.
CGRP antagonist 1 is compound 20[1].
[1]. Stump CA, et al. The discovery of highly potent CGRP receptor antagonists. Bioorg Med Chem Lett. 2009 Jan 1;19(1):214-7.