AS2717638是一种具有口服生物活性的，啮齿动物中溶血磷脂酸受体5(LPA5)的拮抗剂。AS2717638还能增强PGE2、PGF2α以及AMPA诱导的异位疼痛。
货号:ajcx12692
CAS:2148339-28-8
分子式:C25H25N3O5
分子量：447.48
溶解度:Soluble in DMSO
纯度：98%
存储：Store at -20°C
库存：现货

Background:

AS2717638 is an oral active lysophosphatidic acid receptor 5 (LPA5) antagonist in rodents. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia[1].

[1]. Murai N, et al. Analgesic effects of novel lysophosphatidic acid receptor 5 antagonist AS2717638 in rodents. Neuropharmacology. 2017 Nov;126:97-107.