Nicardipine D3 hydrochloride 是 Nicardipine hydrochloride 的氘代物。Nicardipine hydrochloride 是一种钙通道 (calcium channel) 阻滞剂,可阻断心脏钙通道,IC50 为 1 μM。Nicardipine hydrochloride 可用于慢性心绞痛以及控制血压的研究。
货号:ajcx38458
CAS:1432061-50-1
分子式:C26H27D3ClN3O6
分子量:519
溶解度:N/A
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Nicardipine D3 hydrochloride (YC-93 D3) is the deuterium labeled Nicardipine hydrochloride. Nicardipine hydrochloride is a calcium channel blocker with an IC50 of 1 μM for blocking cardiac calcium channels. Nicardipine hydrochloride acts as an agent for chronic stable angina and for controlling blood pressure[1].
[1]. Charnet P, et al. Electrophysiological analysis of the action of nifedipine and nicardipine on myocardial fibers. Fundam Clin Pharmacol. 1987;1(6):413-31.