A tetrapeptide µ-opioid receptor agonist
货号:ajcx21804
CAS:2393865-97-7
分子式:C28H38N4O5
分子量：510.6
溶解度:
纯度：98%
存储：Store at -20°C
库存：
现货Background:
Bilaid A is a tetrapeptide agonist of the μ-opioid receptor (Ki= 3.1 μM using HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation in HEK293 cells expressing the human μ-opioid receptor by 21% when used at a concentration of 10 μM.
1.Dekan, Z., Sianati, S., Yousuf, A., et al.A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptorProc. Natl. Acad. Sci. USA116(44)22353-22358(2019)
