QCA570 is an highly potent and efficacious BET degrader based on PROTAC, with an IC50 of 10 nM for BRD4 BD1 Protein. QCA570 achieves complete and durable tumor regression in leukemia xenograft models in mice at well-tolerated dose-schedules. QCA570 is the most potent and efficacious BET degrader reported to date.
纯度：≥98%
CAS：2207569-08-0
