Paliperidonepalmitate(9-Hydroxyrisperidonepalmitate)是一种非典型长效抗精神病药,是Paliperidone的酯类前药。Paliperidone是一种非典型抗精神病药的多巴胺(dopamine)拮抗剂和5-HT2A拮抗剂。Paliperidonepalmitate对精神分裂症有效。
货号:ajcx31266
CAS:199739-10-1
分子式:C39H57FN4O4
分子量:664.89
溶解度:N/A
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester prodrug of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia[1].
[1]. Kwon JS, et al. Satisfaction of immediate or delayed switch to paliperidone palmitate in patients unsatisfied with current oral atypical antipsychotics. Int Clin Psychopharmacol. 2015;30(6):320-328.