Tasipimidine sulfate 是一种具有口服活性的、选择性的 α2A-adrenoceptor 激动剂,对人 α2A-adrenoceptor 的pEC50 为 7.57。Tasipimidine sulfate 可用于情境焦虑和恐惧的研究。
货号:ajcx39264
CAS:1465908-73-9
分子式:C13H18N2O6S
分子量:330.36
溶解度:DMSO : 125 mg/mL (378.38 mM; ultrasonic and warming and heat to 60°C)
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Tasipimidine sulfate is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 against human α2A-adrenoceptor. Tasipimidine sulfate can be used for situational anxiety and fear research[1].
[1]. LehtimÄki J, et al. Tasipimidine-the pharmacological profile of a novel orally active selective α2A-adrenoceptor agonist. Eur J Pharmacol. 2022 May 15;923:174949.