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ISCK03
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
ISCK03图片
CAS NO:945526-43-2
规格:≥98%
包装与价格:
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ISCK03 is a potent c-kit inhibitor. ISCK03 inhibits SCF/c-kit signaling in 501mel human melanoma cells and abolishes melanin production in mice and brownish guinea pigs. ISCK03 also inhibited p44/42 ERK mitogen-activated protein kinase (MAPK) phosphorylation, which is known to be involved in SCF/c-kit downstream signaling. ISCK03 might be used as skin-whitening agents. References: Na YJ, Baek HS, Ahn SM, Shin HJ, Chang IS, Hwang JS.
[4-t-butylphenyl]-N-(4-imidazol-1-yl phenyl)sulfonamide (ISCK03) inhibits
SCF/c-kit signaling in 501mel human melanoma cells and abolishes melanin
production in mice and brownish guinea pigs. Biochem Pharmacol. 2007 Sep
1;74(5):780-6. Epub 2007 Jun 14. PubMed PMID: 17658483.
 
 
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