α-Terpinyl acetate 是从 Laurus nobilis L. 精油中分离出的一种单萜酯。α-Terpinyl acetate 是竞争性的 P450 2B6 底物，与其活性部位结合的 Kd 值为 5.4 ?μM 。
| Cas No. | 80-26-2 |
| 分子式 | C12H20O2 |
| 分子量 | 196.29 |
| 溶解度 | DMSO : 100 mg/mL (509.45 mM; Need ultrasonic) |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | α-Terpinyl acetate is a monoterpene ester isolated fromLaurus nobilis L.essential oil. α-Terpinyl acetate is a competitiveP450 2B6substrate which binding to the active site of P450 2B6 with aKdvalue of 5.4?μM[1][2]. The bupropion hydroxylation activity of P450 2B6 is inhibited by α-Terpinyl acetate wiht an IC50value of 10.4?μM and α-Terpinyl acetate is determined to be a competitive inhibitor of P450 2B6 with a Kiof 7.6 ?μM[2].
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