Dazcapistat 是一种有效的钙蛋白酶 (calpain) 抑制剂,对 calpain 1, calpain 2 和calpain 9 的 IC50 值为<3 μM (详细信息请参见专利WO2018064119A1, compound 405)。
Cas No. | 2221010-42-8 |
分子式 | C21H18FN3O4 |
分子量 | 395.38 |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Dazcapistat is a potent calpain inhibitor, with IC50s of<3 μM for calpain 1, calpain 2 and calpain 9, respectively (patent WO2018064119A1, compound 405)[1]. [1]. Brad Owen BUCKMAN, et al. Calpain modulators and therapeutic uses thereof. WO2018064119A1. |