首页 蛋白库 基因库 产品 会员服务
位置：首页 > 产品库 > Adenosine receptor antagonist 2
立即咨询
咨询类型：
     
*姓名：
*电话：
*单位：
Email：
*留言内容：
请详细说明您的需求。
*验证码：
 
Adenosine receptor antagonist 2
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Adenosine receptor antagonist 2图片
CAS NO:2703054-47-9
包装:10mg
市场价:11250元

Adenosine receptor antagonist 2 是一种口服有效的 A2a/A2b 腺苷受体拮抗剂，IC50 分别为 1 nM 和 3 nM。Adenosine receptor antagonist 2 具有抗肿瘤活性。
Cas No.2703054-47-9
分子式C23H21FN8O
分子量444.46
储存条件4°C, away from moisture and light
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Adenosine receptor antagonist 2 is an orally activeA2a/A2b adenosine receptorantagonist withIC50s of 1 nM and 3 nM, respectively. Adenosine receptor antagonist 2 has anti-tumor activity[1].

Adenosine receptor antagonist 2 (compound L-1; po; 10, 30, 100 mg/kg; twice a day for 22 days) inhibits tumor growth in female C57BL / 6mice mice with MC38(#22)-hpd-L1 cells[1].
Adenosine receptor antagonist 2 (iv; 2 mg/kg) has a CLz of 14.7 mL/min.kg and an AUC of 2252 h.ng/mL. Adenosine receptor antagonist 2 (po; 10 mg/kg) has a Cmaxof 8730 ng/mL in adult male ICR mice (weight 25-40g)[1].

 
 
维奥蛋白资源库 - 中文蛋白资源 CopyRight © 2010-2024