Enzalutamide D3 是一种氘标记的 Enzalutamide (MDV3100)。Enzalutamide 是一种雄激素受体 (AR) 拮抗剂,在 LNCaP 前列腺细胞中 IC50 为 36 nM。
Cas No. | 1443331-82-5 |
别名 | 恩杂鲁胺-D3,Enzalutamide-d3; MDV3100-d3 |
分子式 | C21H13D3F4N4O2S |
分子量 | 467.45 |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Enzalutamide D3 is a deuterium labeled Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells[1]. [1]. Tran C, et al. Development of a second-generation antiandrogen for treatment of advanced prostate cancer. Science. 2009 May 8;324(5928):787-90. |