RY796 是一种有效的选择性电压门控钾 (KV2) 通道抑制剂,对 KV2.1 和 KV2.2 的 IC50 值分别为 0.25 μM 和 0.09 μM。RY796 可用于缓解疼痛的研究。
Cas No. | 1393441-53-6 |
分子式 | C21H27N3O2 |
分子量 | 353.46 |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | RY796 is a potent and selective voltage-gated potassium (KV2) channel inhibitor with IC50s of 0.25 μM and 0.09 μM for KV2.1 and KV2.2. RY796 has analgesic activity[1]. [1]. Herrington J, et al. Identification of novel and selective Kv2 channel inhibitors. Mol Pharmacol. 2011 Dec;80(6):959-64. |