TRPM8 antagonist 3 是一种新型的 TRPM8 阻滞剂,其 IC50 值为 11 nM。
Cas No. | 2102179-29-1 |
分子式 | C13H12N2O4S |
分子量 | 292.31 |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | TRPM8 antagonist 3 is a novel TRPM8 blocker with an IC50 value of 11 nM. [1]. Bianchini G, et al. Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions: A Journey through pKa and LogD Modulation. J Med Chem. 2021 Nov 25;64(22):16820-16837. |