(R)-Funapide ((R)-TV 45070) 是 Funapide 活性较低的 R-对映异构体。Funapide 是一种有效的 Nav1.7 钠通道阻滞剂,可用于疼痛研究。
Cas No. | 1259933-15-7 |
别名 | (R)-TV 45070; (R)-XEN402 |
分子式 | C22H14F3NO5 |
分子量 | 429.35 |
溶解度 | DMSO : 220 mg/mL (512.40 mM; Need ultrasonic) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | (R)-Funapide ((R)-TV 45070) is the less active R-enantiomer of Funapide. Funapide is a potent Nav1.7 sodium channel blocker that can be used for pain research[1]. [1]. Sharan K Bagal, et al. Recent progress in sodium channel modulators for pain. Bioorg Med Chem Lett. 2014 Aug 15;24(16):3690-9. |