Bopindolol ((±)-Bopindolol) malonate 是 β-adrenoceptors (ARs) 的口服活性拮抗剂,具有部分激动剂活性。
Cas No. | 82857-38-3 |
别名 | (±)-Bopindolol (malonate) |
Canonical SMILES | O=C(O)CC(O)=O.O=C(OC(COC1=CC=CC2=C1C=C(C)N2)CNC(C)(C)C)C3=CC=CC=C3 |
分子式 | C23H28N2O3•C3H4O4 |
分子量 | 484.5 |
溶解度 | Water: 5mM |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Bopindolol is a non-selective β-adrenergic receptor antagonist. In vivo, bopindolol decreases heart rate and blood pressure and attenuates ischemia-induced myocardial acidosis in dogs. Formulations containing bopindolol have been used to treat essential and renovascular hypertension. |