ent-LP 99 是一种有效的选择性 BRD7 和 BRD9 抑制剂，对 BRD9 的 KD 为 99 nM。
| Cas No. | 1808948-28-8 |
| Canonical SMILES | CC(C(C=C1)=C(N2C)C=C1N3[C@@H](C4=CC=C(Cl)C=C4)[C@H](NS(=O)(CC(C)C)=O)CCC3=O)=CC2=O |
| 分子式 | C26H30ClN3O4S |
| 分子量 | 516.05 |
| 溶解度 | Soluble in DMSO |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Negative Control for LP 99 (Cat.No. 5496). Clark et al (2015) LP99: discovery and synthesis of the first selective BRD7/9 bromodomain inhibitor. Angew.Chem.Int.Ed.Engl. 54 6217 PMID:25864491 |
