(rac)-BAY1238097是一种BET抑制剂，对BRD4的IC50值为1.02μM。用于癌症研究。
| Cas No. | 1564268-19-4 |
| Canonical SMILES | CC1N(C(NC)=O)N=C(C2=CC=C(N3CCN(C)CC3)C=C2)C4=CC(OC)=C(OC)C=C4C1 |
| 分子式 | C25H33N5O3 |
| 分子量 | 451.56 |
| 溶解度 | DMSO : 150 mg/mL (332.18 mM) |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | (rac)-BAY1238097 is a BET inhibitor, with an IC50 of 1.02 μM for BRD4. Used in cancer research[1].
IC50: 1.02 μM (BRD4)[1] [1]. Stephan Siegel, et al. 2,3-benzodiazepines. WO2014026997A1. |
