CP-409092 hydrochloride 是 GABAA 受体的部分激动剂,具有抗焦虑活性。
Cas No. | 225240-86-8 |
Canonical SMILES | O=C(C1=CNC2=C1C(CCC2)=O)NC3=CC=C(CNC)C=C3.Cl |
分子式 | C17H20ClN3O2 |
分子量 | 333.81 |
溶解度 | DMSO: 41.67 mg/mL (124.83 mM) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity[1]. [1]. Kamel A, et al. Metabolism, pharmacokinetics and excretion of the GABA(A) receptor partial agonist [(14)C]CP-409,092 in rats. Xenobiotica. 2010 Jun;40(6):400-14. |