PL 017 是一种有效的选择性 μ 阿片受体激动剂，125I-FK 33,824 与 μ 位点结合的 IC50 为 5.5 nM。
| Cas No. | 83397-56-2 |
| 别名 | N-Me-phe（3）-吗啡肽 |
| 化学名 | (S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N-((S)-1-((R)-2-carbamoylpyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-N-methylpyrrolidine-2-carboxamide |
| Canonical SMILES | O=C([C@H]1N(C([C@H](CC(C=C2)=CC=C2O)N)=O)CCC1)N(C)[C@@H](CC3=CC=CC=C3)C(N4[C@@H](C(N)=O)CCC4)=O |
| 分子式 | C29H37N5O5 |
| 分子量 | 535.64 |
| 溶解度 | Soluble to 1 mg/ml in Water |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
