Taranabant (1R，2R)stereoisomer 是 Taranabant 的 R 型对映异构体。Taranabant 是有效的选择性 cannabinoid 1 (CB1) 受体反向激动剂。
| Cas No. | 701977-08-4 |
| 别名 | MK0364 (1R,2R)stereoisomer |
| Canonical SMILES | CC(OC1=NC=C(C(F)(F)F)C=C1)(C)C(N[C@H](C)[C@@H](C2=CC=CC(C#N)=C2)CC3=CC=C(Cl)C=C3)=O |
| 分子式 | C27H25ClF3N3O2 |
| 分子量 | 515.95 |
| 溶解度 | DMSO: 100 mg/mL (193.82 mM); Water:< 0.1 mg/mL (insoluble) |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. [1]. William K. Hagmann, et al. Substituted amides active at the cannabinoid-1 receptor. WO 2004048317 A1. |
