| CAS NO: | 1893-33-0 |
| Cas No. | 1893-33-0 |
| 别名 | 酰胺哌啶酮,Floropipamide; McN-JR 3345; R 3345 |
| Canonical SMILES | O=C(C1(N2CCCCC2)CCN(CCCC(C3=CC=C(F)C=C3)=O)CC1)N |
| 分子式 | C21H30FN3O2 |
| 分子量 | 375.48 |
| 溶解度 | 0.1 M HCL: 25 mg/mL (66.58 mM) |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | Pipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7)[1]. 5-HT2A Receptor|8.2 (pKi)|5-HT2C Receptor|6.9 (pKi)|5-HT1 Receptor|5.7 (pKi)|D4 receptor|8.0 (pKi)|D2 receptor|6.7 (pKi)|α1 receptor|7.2 (pKi) [1]. Erik Buntinx, MD, et al. Selective Serotonergic Properties of Low-Dose Pipamperone May Enhance Antidepressant Effect: Preclinical Evidence. |
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