CAS NO: | 1008763-54-9 |
包装 | 价格(元) |
10mM (in 1mL DMSO) | 询价 |
1mg | 询价 |
5mg | 询价 |
10mg | 询价 |
50mg | 询价 |
100mg | 询价 |
Cas No. | 1008763-54-9 |
Canonical SMILES | [H]Cl.O=C1N(CCN)C2=CC(OC)=CC=C2N1C([C@H]3[C@H](C(C)C)CC[C@@H](C)C3)=O |
分子式 | C21H32ClN3O3 |
分子量 | 409.95 |
溶解度 | DMSO : ≥ 40 mg/mL (97.57 mM) |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | D-3263 hydrochloride is an enteric-coated, orally bioavailable (transient receptor potential melastatin member 8) TRPM8 agonist. D-3263 hydrochloride binds to and activates TRPM8, which may result in an increase in calcium and sodium entry; the disruption of calcium and sodium homeostasis; and the induction of cell death in TRPM8-expressing tumor cells. D-3263 hydrochloride may decrease dihydrotestosterone (DHT) levels, which may contribute to its inhibitory effects on prostate cancer and BPH[1]. [1]. enteric-coated TRPM8 agonist D-3263 hydrochloride |
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