Nevanimibe hydrochloride(PD-132301 hydrochloride ATR101 hydrochloride)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
| CAS: | 133825-81-7 |
| 分子式: | C27H40ClN3O |
| 分子量: | 458.08 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | ACAT1; 9 nM (EC50); ACAT2; 368 nM (EC50) |
| 描述: | Nevanimibe hydrochloride is a selective, potent acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) inhibitor with an EC50 of 9 nM. Nevanimibe hydrochlorid inhibits ACAT2 with an EC50 of 368 nM. |