Lonafarnib(Sch66336)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
| 产品名称: | 洛那法尼 |
| CAS: | 193275-84-2 |
| 分子式: | C27H31Br2ClN4O2 |
| 分子量: | 638.82 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | IC50: 1.9 nM (H-ras), 5.2 nM (K-ras), 2.8 nM (N-ras)[1] |
| 描述: | Lonafarnib is an orally bioavailable farnesyl protein transferase (FPTase) inhibitor for H-ras, K-ras and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM, respectively. |