BMS-687453
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
包装与价格:
| 包装 | 价格(元) |
| 5mg | 询价 |
| 10mg | 询价 |
| 50mg | 询价 |
| 100mg | 询价 |
| CAS: | 1000998-59-3 |
| 分子式: | C22H21ClN2O6 |
| 分子量: | 444.86 |
| 纯度: | ≥98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cardiovascular disease |
| Target: | EC50: 10 nM (GAL4-human PPARα), 4100 nM (GAL4-human PPARγ)[1]IC50: 260 nM (Human PPARα), >15000 nM (Human PPARγ)[1] |
| 描述: | BMS-687453 is a potent and selective PPARα agonist, with an EC50 and IC50 of 10 nM and 260 nM for human PPARα and 4100 nM and >15000 nM for PPARγ in PPAR-GAL4 transactivation assays. |