| CAS： | 1936421-41-8 |
| 分子式： | C27H32F2N6O2 |
| 分子量： | 510.58 |
| 纯度： | >98% |
| 溶解性： | DMSO |
| 存储： | -20℃, stored under nitrogen. In solvent : -80℃, 6 months; -20℃, 1 month (stored under nitrogen) |
| 研究领域： | Cancer |
| Target： | IC50: 1.1 nM (CBP), 12 nM (BRET), 4200 nM (BRD4(1)) |
| 描述： | GNE-049 is a highly potent and selective CBP inhibitor with an IC50 of 1.1 nM in TR-FRET assay. GNE-049 also inhibits BRET and BRD4(1) with IC50s of 12 nM and 4200 nM, respectively. |
