TAK-632
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
包装与价格:
| 包装 | 价格(元) |
| 10mg | 询价 |
| 50mg | 询价 |
| 100mg | 询价 |
| CAS: | 1228591-30-7 |
| 分子式: | C27H18F4N4O3S |
| 分子量: | 554.52 |
| 纯度: | >98% |
| 溶解性: | DMSO |
| 存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
| 研究领域: | Cancer |
| Target: | 1.4 nM (IC50)-c-Raf,8.3 nM (IC50)-Braf,66 nM (IC50)-Aurora B,120 nM (IC50)-PDGFRβ,610 nM (IC50)-PDGFRα,280 nM (IC50)-FGFR3,740 nM (IC50)-TIE2,3700 nM (IC50)-IKKβ,790 nM (IC50)-CDK1,580 nM (IC50)-CDK2, |
| 描述: | TAK-632 is a potent pan-RAF inhibitor with IC50 of 1.4, 2.4 and 8.3 nM for CRAF, BRAFV600E, BRAFWT, respectively. |