TRPVantagonist1是一种有效的瞬时受体电位V型(TRPV)拮抗剂,IC50值<250nM。
Cas No. | 1192871-27-4 |
Canonical SMILES | O=C1C(C2=CC=C(OC(F)(F)F)C=C2)=C(/C=C/C3=CC=CC(OC)=C3OCC4CC4)N=C5N1C=CS5 |
分子式 | C26H21F3N2O4S |
分子量 | 514.52 |
溶解度 | Soluble in DMSO |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | TRPV antagonist 1 is a transient receptor potential vanilloid (TRPV) antagonist, with an IC50 of< 250 nM. [1]. Reilly RM, et al. Analgesic potential of TRPV3 antagonists. Curr Top Med Chem. 2011;11(17):2210-5. |