Beperidium iodide (SX 810) 对乙酰胆碱受体具有竞争性拮抗作用,pA2 为 7.93。
Cas No. | 86434-57-3 |
别名 | 贝哌碘铵,SX 810 |
Canonical SMILES | C[N+]1(CC)CCC(OC(C(C2=NOC3=C2C=CC=C3)N4CCCCCC4)=O)CC1.[I-] |
分子式 | C23H34IN3O3 |
分子量 | 527.44 |
溶解度 | Soluble in DMSO |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | Beperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93. [1]. Kawashima K, et al. Pharmacological properties of the novel antimuscarinic agent 4-[2-(1,2-benzisoxazol-3-yl)-2-(hexahydro-1H-azepin-1-yl)a cetoxy]-1-et hyl-1- methylpiperidinium iodide. Arzneimittelforschung. 1986 Jun;36(6):927-35. |