EP1-antanoist-1 是一种 EP1 拮抗剂，pKi 为 7.54，pIC50 为 8.5。
| Cas No. | 851204-35-8 |
| Canonical SMILES | O=C(C1=NN(CC2=CC(Br)=CC=C2OCC3=CC=C(Cl)C=C3Cl)C(C)=C1)O |
| 分子式 | C19H15BrCl2N2O3 |
| 分子量 | 470.14 |
| 溶解度 | Soluble in DMSO |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | EP1-antanoist-1 is a EP1 antagonist with a pKi of 7.54 and an pIC50 of 8.5. [1]. McKeown SC, et al. Identification of novel pyrazole acid antagonists for the EP1 receptor. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4767-71. Epub 2006 Jul 14. |
