| CAS NO: | 786686-79-1 |
| 包装: | 5mg |
| 市场价: | 9000元 |
| 生物活性 | Olanzapine-d3 (LY170053-d3) is the deuterium labeled Olanzapine. Olanzapine is a selective, orally active monoaminergic antagonist with high affinity binding toserotonin H1, 5HT2A/2C, 5HT3, 5HT6(Ki=7, 4, 11, 57, and 5 nM, respectively),dopamine D1-4(Ki=11 to 31 nM),muscarinic M1-5(Ki=1.9-25 nM), andadrenergic α1 receptors(Ki=19 nM). Olanzapine is an atypical antipsychotic[1][2]. | ||||||||||||
| IC50& Target |
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| 分子量 | 315.45 | ||||||||||||
| 性状 | Solid | ||||||||||||
| Formula | C17H17D3N4S | ||||||||||||
| CAS 号 | 786686-79-1 | ||||||||||||
| 中文名称 | 奥氮平 d3;奥兰氮平 d3 | ||||||||||||
| 运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| 储存方式 |
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