APJ receptor agonist 6 (compound 9) 是一种有效的APJ(apelin 受体)激动剂，其Ki为 0.059 μM。APJ receptor agonist 6 对钙 (calcium)、cAMP和β-arrestin的EC50分别为 0.800、0.844 和 6.22 μM。
| 生物活性 | APJ receptor agonist 6 (compound 9) is a potentAPJ(apelin receptor) agonist, withKiof 1.3 μM. APJ receptor agonist 6 hasEC50values of 0.070 , 0.097, and 0.063 μM forcalcium,cAMP, andβ-arrestin, respectively[1]. |
| IC50& Target | EC50: 0.800 ± 0.1 μM (Apelin Receptor calcium), 0.844 ± 0.2 μM (Apelin Receptor cAMP), 6.22 ± 2.0 μM (Apelin Receptor β-arrestin), >10 μM (AT1 calcium)[1] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
