GRK2i 是一种Gβγ抑制肽,可选择性地阻止 Gβγ 介导的信号传导。GRK2i 对应于 GRK2(G 蛋白偶联受体激酶 2)的 Gβγ 结合域。
生物活性 | GRK2i is aGβγ-inhibitory peptide that selectively prevents Gβγ-mediated signaling. GRK2i corresponds to the Gβγ-binding domain of GRK2 (G-protein-coupled receptor kinase 2)[1]. |
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体外研究 (In Vitro) | GRK2i (5 μM) inhibits neurite formation, disrupts microtubules, and induces neurite damag in PC12 cells[1].
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Sequence Shortening | WKKELRDAYREAQQLVQRVPKMKNKPRS |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |