RSK2-IN-2

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RSK2-IN-2

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

1637749-78-0

RSK2-IN-2 (Compound 25) 是 RPS6KA3 (RSK2) 激酶的可逆共价抑制剂。 RSK2-IN-2 也抑制MSK1、MSK2和RSK3。

生物活性

RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 (RSK2) kinase. RSK2-IN-2 is also described to inhibitMSK1,MSK2andRSK3^[1].

IC₅₀& Target

RSK2

RSK3

MSK1

MSK2

体外研究
(In Vitro)

RSK2-IN-2 (Compound 25) shows strong activity with ERK2-MSK1 cascade pIC₅₀of 9.6^[1].

分子量

289.29

Formula

C₁₆H₁₁N₅O

CAS 号

1637749-78-0

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.