MEDICA16 是一种ATP-citrate lyase抑制剂，能显著降低腓肠肌细胞内 TG 的含量，这种降低伴随着胰岛素敏感性的增加。MEDICA16 是GPR40的选择性激动剂，也是GPR120的选择性部分激动剂。
| 生物活性 | MEDICA16, anATP-citrate lyaseinhibitor, significantly reduces intracellular TG content in gastrocnemius muscle, and this reduction is accompanied by an increase ininsulinsensitivity. MEDICA16 is a selective agonist forGPR40as well as selective partial agonists forGPR120[1][2]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Pure form | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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