CETP-IN-3

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CETP-IN-3

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CAS NO:

939391-31-8

CETP-IN-3 (Compound 13) 是血浆糖蛋白胆固醇酯转移蛋白 (CETP) 的小分子抑制剂，可抑制 CETP 活性并提高高密度脂蛋白胆固醇 (HDL-C) 水平。CETP-IN-3 抑制活力的IC₅₀值分别为0.002 μM (SPA), 0.06 μM (WPA) 。

生物活性	CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasmaglycoproteincholesterol ester transfer protein (CETP), elevating HDL-C through inhibition ofCETP. CETP-IN-3 for theCETPinhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) withIC₅₀s of 0.002 μM and 0.06 μM, respectively^[1].
分子量	704.50
Formula	C₃₀H₂₄F₁₂N₂O₄
CAS 号	939391-31-8
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.