EphA2 agonist 1 (Compound 7bg) 是一种有效的EphA2 receptor激动剂。EphA2 agonist 1 对 EphA2 过表达的胶质瘤细胞具有很强的活性和选择性,并能刺激EphA2磷酸化。
生物活性 | EphA2agonist 1 (Compound 7bg) is a potentEphA2receptoragonist.EphA2agonist 1 shows great potency and selectivity towardEphA2overexpressed glioblastoma cells and stimulatesEphA2phosphorylation[1]. |
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体外研究 (In Vitro) | EphA2 agonist 1 (Compound 7bg) inhibits cell proliferation with IC50values of 1.90 ± 0.55 μM and 7.91 ± 2.28 μM against U251 EphA2 overexpressed and U251 wild type cells, respectively[1].
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |