CGP 54626 (hydrochloride) 是 GABAB 受体的选择性拮抗剂,IC50 值为 4 nM。
Cas No. | 149184-21-4 |
别名 | TOCCGP54626盐酸盐 |
化学名 | (S)-(cyclohexylmethyl)((S)-3-(((S)-1-(3,4-dichlorophenyl)ethyl)amino)-2-hydroxypropyl)phosphinic acid hydrochloride |
Canonical SMILES | ClC1=CC([C@H](C)NC[C@@H](C[P@@](O)(CC2CCCCC2)=O)O)=CC=C1Cl.Cl |
分子式 | C18H28Cl2NO3P.HCl |
分子量 | 444.76 |
溶解度 | DMF: 0.33 mg/ml,DMSO: 1 mg/ml,DMSO:PBS (pH 7.2) (1:6): 0.14 mg/ml,Ethanol: 0.2 mg/ml |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |