| CAS NO: | 113-79-1 |
| 生物活性 | Argipressin (Arg8-vasopressin) binds to theV1, V2, V3-vascular argininevasopressin receptor, with aKdvalue of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1. | ||||||||||||||||
| IC50& Target |
| ||||||||||||||||
| 体外研究 (In Vitro) | Argipressin binds to the vascular arginine vasopressin receptor, V1, with a Kdvalue of 1.31 nM in A7r5 rat aortic smooth muscle cells. It also stimulates the intracellular release of calcium in A7r5 cells (EC50=5 nM)[1]. AVP-induced [Ca2+]isignals and immunized activity against S-100 in DRG cell culture. The minimum effective concentrations of Argipressin causing [Ca2+]iresponses are 100 pM in non-neuronal cells in DRG culture[2]. | ||||||||||||||||
| Clinical Trial | |||||||||||||||||
| 分子量 | 1084.23 | ||||||||||||||||
| 性状 | Solid | ||||||||||||||||
| Formula | C46H65N15O12S2 | ||||||||||||||||
| CAS 号 | 113-79-1 | ||||||||||||||||
| Sequence | Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: Cys1-Cys6) | ||||||||||||||||
| Sequence Shortening | CYFQNCPRG-NH2 (Disulfide bridge: Cys1-Cys6) | ||||||||||||||||
| 中文名称 | 精氨加压素 | ||||||||||||||||
| 运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
| 储存方式 | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||||||||||||
| 溶解性数据 | In Vitro: H2O : ≥ 100 mg/mL(92.23 mM) *"≥" means soluble, but saturation unknown. 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
| 维奥蛋白资源库 - 中文蛋白资源 CopyRight © 2010-2026 |
