P2X7-IN-2 (compound 58) 是P2X7受体抑制剂。P2X7-IN-2 抑制 IL-Iβ 的释放,IC50值为 0.01 nM。P2X7-IN-2 可用于自身免疫病,炎症以及心血管疾病的研究。
生物活性 | P2X7-IN-2 (compound 58) is aP2X7receptor inhibitor. P2X7-IN-2 inhibits IL-Iβ release with anIC50value of 0.01 nM. P2X7-IN-2 can be used for the research of autoimmunity, inflammation andcardiovascular disease[1]. |
IC50& Target | IC50: 0.01 nM (human whole blood IL-Iβ release)[1] |
体外研究 (In Vitro) | P2X7-IN-2 (0-1 μM;30 min) inhibits human whole blood IL-Iβ release with an IC50value of 0.01 nM[1].
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |