AK-IN-1 (化合物 4072-2732) 是一种对腺苷 (Ado) 有竞争性但对 ATP 无竞争性的腺苷激酶 (AK) 抑制剂。AK-IN-1 浓度为 2, 4, 10 μM 时，能分别抑制 86%、87% 和 89% 的AK活性。AK-IN-1 在许多疾病领域 (包括缺血、炎症和癫痫发作) 都具有较好的研究潜力。
| 生物活性 | AK-IN-1 (compound 4072-2732) is anadenosine kinase(AK) inhibitor that is competitive for adenosine (Ado) but not for ATP. AK-IN-1 inhibits 86%, 87% and 89% ofAKactivity at concentrations of 2, 4 and 10 μM, respectively. AK-IN-1 has good potential for research in many disease areas, including ischaemia, inflammation and seizures[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
