PDHK-IN-5 (Compound 19) 是一种有效的PDHK抑制剂，对 PDHK2 和 PDHK4 的IC50s 分别为 0.006 和 0.0329 μM。丙酮酸脱氢酶激酶 (PDHK) 是许多疾病（包括糖尿病和癌症）的迷人药物靶点。PDHK-IN-5 具有研究癌症疾病的潜力。
| 生物活性 | PDHK-IN-5 (Compound 19) is a potent inhibitor ofPDHKwithIC50s of 0.006 and 0.0329 μM for PDHK2 and PDHK4, repectively. Pyruvate dehydrogenase kinases (PDHKs) are fascinating drug targets for numerous diseases, including diabetes and cancers. PDHK-IN-5 has the potential for the research ofcancerdiseases[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
