(1S,3R)-GNE-502 (compound 179) 是一种有效的 ERα 降解剂,在 MCF7 HCS 细胞中降解 ERα 的 EC50 为 13 nM。(1S,3R)-GNE-502 可用于研究与雌激素受体相关的癌症。
Cas No. | 1953134-15-0 |
分子式 | C25H30FN3O3S |
分子量 | 471.59 |
储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | (1S,3R)-GNE-502 (compound 179) is a potentERαdegrader with anEC50value of 13 nM against ERα in MCF7 HCS. (1S,3R)-GNE-502 can be used to research cancer related with estrogen receptor[1]. |