H2L5186303 是一种有效的选择性 LPA2 受体（溶血磷脂酸 2 受体）拮抗剂，IC50 为 9 nM。
| Cas No. | 139262-76-3 |
| 化学名 | (2Z,2'Z)-4,4'-(((1,3-phenylenebis(oxy))bis(4,1-phenylene))bis(azanediyl))bis(4-oxobut-2-enoic acid) |
| Canonical SMILES | O=C(NC1=CC=C(OC2=CC(OC3=CC=C(NC(/C([H])=C([H])\C(O)=O)=O)C=C3)=CC=C2)C=C1)/C([H])=C([H])\C(O)=O |
| 分子式 | C26H20N2O8 |
| 分子量 | 488.45 |
| 溶解度 | DMF: 20 mg/mL,DMF:PBS (pH 7.2) (1:8): 0.11 mg/mL,DMSO: 15 mg/mL |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
