CHK1-IN-4 (化合物3) 是一种有效的关卡激酶 1 (chk1) 抑制剂,可有效抑制肿瘤细胞中 chk1 磷酸化。CHK1-IN-4 具有抗肿瘤活性。
生物活性 | CHK1-IN-4 (Compound 3) is a potentcheckpoint kinase 1 (chk1)inhibitor, and potently inhibitschk1phosphorylation in the tumor cells. CHK1-IN-4 has anti-tumor activity[1]. |
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体内研究 (In Vivo) | CHK1-IN-4 (Compound 3) (40 mg/kg, IV, twice a week) alone enhances anti-tumor growth activity of CPT1 in the tumor model[1].
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |